Details for: UGT1A8

Gene ID: 54576

Symbol: UGT1A8

Ensembl ID: ENSG00000242366

Description: UDP glucuronosyltransferase family 1 member A8

Associated with

Other Information

Genular Protein ID: 3024977555

Symbol: UD18_HUMAN

Name: UDP-glucuronosyltransferase 1-8

UniProtKB Accession Codes:

Database IDs:

Citations:

PubMed ID: 9535849

Title: Expression of the UDP-glucuronosyltransferase 1A locus in human colon. Identification and characterization of the novel extrahepatic UGT1A8.

PubMed ID: 9535849

DOI: 10.1074/jbc.273.15.8719

PubMed ID: 11434514

Title: Thirteen UDP-glucuronosyltransferase genes are encoded at the human UGT1 gene complex locus.

PubMed ID: 11434514

DOI: 10.1097/00008571-200106000-00011

PubMed ID: 12042666

Title: Identification and functional characterization of UDP-glucuronosyltransferases UGT1A8*1, UGT1A8*2 and UGT1A8*3.

PubMed ID: 12042666

DOI: 10.1097/00008571-200206000-00004

PubMed ID: 14702039

Title: Complete sequencing and characterization of 21,243 full-length human cDNAs.

PubMed ID: 14702039

DOI: 10.1038/ng1285

PubMed ID: 15815621

Title: Generation and annotation of the DNA sequences of human chromosomes 2 and 4.

PubMed ID: 15815621

DOI: 10.1038/nature03466

PubMed ID: 12181437

Title: Common human UGT1A polymorphisms and the altered metabolism of irinotecan active metabolite 7-ethyl-10-hydroxycamptothecin (SN-38).

PubMed ID: 12181437

DOI: 10.1124/mol.62.3.608

PubMed ID: 15472229

Title: Specificity and regioselectivity of the conjugation of estradiol, estrone, and their catecholestrogen and methoxyestrogen metabolites by human uridine diphospho-glucuronosyltransferases expressed in endometrium.

PubMed ID: 15472229

DOI: 10.1210/jc.2004-0331

PubMed ID: 15470161

Title: Identification of the UDP-glucuronosyltransferase isoforms involved in mycophenolic acid phase II metabolism.

PubMed ID: 15470161

DOI: 10.1124/dmd.104.001651

PubMed ID: 16595710

Title: Human UDP-glucuronosyltransferase, UGT1A8, glucuronidates dihydrotestosterone to a monoglucuronide and further to a structurally novel diglucuronide.

PubMed ID: 16595710

DOI: 10.1124/dmd.106.009621

PubMed ID: 17179145

Title: Oligomerization of the UDP-glucuronosyltransferase 1A proteins: homo- and heterodimerization analysis by fluorescence resonance energy transfer and co-immunoprecipitation.

PubMed ID: 17179145

DOI: 10.1074/jbc.m609417200

PubMed ID: 18052087

Title: Disposition of flavonoids via enteric recycling: enzyme stability affects characterization of prunetin glucuronidation across species, organs, and UGT isoforms.

PubMed ID: 18052087

DOI: 10.1021/mp700135a

PubMed ID: 18004212

Title: Genetic diversity at the UGT1 locus is amplified by a novel 3' alternative splicing mechanism leading to nine additional UGT1A proteins that act as regulators of glucuronidation activity.

PubMed ID: 18004212

DOI: 10.1097/fpc.0b013e3282f1f118

PubMed ID: 18674515

Title: The human UDP-glucuronosyltransferase UGT1A3 is highly selective towards N2 in the tetrazole ring of losartan, candesartan, and zolarsartan.

PubMed ID: 18674515

DOI: 10.1016/j.bcp.2008.07.006

PubMed ID: 18719240

Title: The configuration of the 17-hydroxy group variably influences the glucuronidation of beta-estradiol and epiestradiol by human UDP-glucuronosyltransferases.

PubMed ID: 18719240

DOI: 10.1124/dmd.108.022731

PubMed ID: 19159218

Title: Glycoproteomics analysis of human liver tissue by combination of multiple enzyme digestion and hydrazide chemistry.

PubMed ID: 19159218

DOI: 10.1021/pr8008012

PubMed ID: 19545173

Title: Structure and concentration changes affect characterization of UGT isoform-specific metabolism of isoflavones.

PubMed ID: 19545173

DOI: 10.1021/mp8002557

PubMed ID: 20610558

Title: Alternatively spliced products of the UGT1A gene interact with the enzymatically active proteins to inhibit glucuronosyltransferase activity in vitro.

PubMed ID: 20610558

DOI: 10.1124/dmd.110.034835

PubMed ID: 23288867

Title: Regiospecificity and stereospecificity of human UDP-glucuronosyltransferases in the glucuronidation of estriol, 16-epiestriol, 17-epiestriol, and 13-epiestradiol.

PubMed ID: 23288867

DOI: 10.1124/dmd.112.049072

PubMed ID: 19204906

Title: Analysis of inherited genetic variations at the UGT1 locus in the French-Canadian population.

PubMed ID: 19204906

DOI: 10.1002/humu.20946

Sequence Information:

  • Length: 530
  • Mass: 59742
  • Checksum: AD838436940F4190
  • Sequence:
  • MARTGWTSPI PLCVSLLLTC GFAEAGKLLV VPMDGSHWFT MQSVVEKLIL RGHEVVVVMP 
    EVSWQLGKSL NCTVKTYSTS YTLEDLDREF MDFADAQWKA QVRSLFSLFL SSSNGFFNLF 
    FSHCRSLFND RKLVEYLKES SFDAVFLDPF DACGLIVAKY FSLPSVVFAR GIACHYLEEG 
    AQCPAPLSYV PRILLGFSDA MTFKERVRNH IMHLEEHLFC QYFSKNALEI ASEILQTPVT 
    AYDLYSHTSI WLLRTDFVLD YPKPVMPNMI FIGGINCHQG KPLPMEFEAY INASGEHGIV 
    VFSLGSMVSE IPEKKAMAIA DALGKIPQTV LWRYTGTRPS NLANNTILVK WLPQNDLLGH 
    PMTRAFITHA GSHGVYESIC NGVPMVMMPL FGDQMDNAKR METKGAGVTL NVLEMTSEDL 
    ENALKAVIND KSYKENIMRL SSLHKDRPVE PLDLAVFWVE FVMRHKGAPH LRPAAHDLTW 
    YQYHSLDVIG FLLAVVLTVA FITFKCCAYG YRKCLGKKGR VKKAHKSKTH

Database document:

This is a preview of the gene's schema. Only a few entries are kept for 'singleCellExpressions,' 'mRNAExpressions,' and other large data arrays for visualization purposes. You can zoom in with the mouse wheel for a closer view, and the text will adjust automatically if necessary. For the full schema, download it here.